Latest Publications

 

1. Kamal Sweidan, Jörn Engelmann, Walid Abu Rayyan, Dima Sabbah, Musa Abu Zarga, Tariq Al-Qirim,Yusuf Al-Hiari, Ghassan Abu Sheikha, Ghassan Shattat. Synthesis and Preliminary Biological Evaluation of New Heterocyclic Carboxamide Models. LDDD, 2014, accepted and in press.

http://benthamscience.com/journal/abstracts.php?journalID=lddd&articleID=126527

 

2. Al-Qirim, Tariq; Shattat, Ghassan; Abu Sheikha, Ghassan; Sweidan, Kamal; Al-Hiari, Yusuf; Jarab, Anan. Synthesis and in vivo antihyperlipidemic activity of new series of N-(4-benzoylphenyl)-2-furamide derivatives Triton-WR-1339-Induced hyperlipidemic Rats. Drug Research, 2014, accepted and in press.

http://www.unboundmedicine.com/medline/citation/24848001/

 

3. Manal AL-Najdawi, Yusuf Al-Hiari, Tariq Al-Qirim, Ghassan Shattat, Mohammad Al-Zweri and Ghassan Abu Sheikha.  Synthesis and Pharmacological Evaluation of Novel Unsubstituted Indole-Anthraquinone Carboxamides Derivatives as Potent Anti-hyperlipidemic Agents. Z. Naturforsch, 69c. 2014, 21-28.

http://www.znaturforsch.com/ac/v69c/69c0021.htm

 

4. Reema Abu Khalaf, Ghassan Abu Sheikha, Mahmoud Al-Sha’er, Mutasem Taha. Design, Synthesis and Biological Evaluation of N4-Sulfonamido-Succinamic, Phthalamic, Acrylic and Benzoyl Acetic Acid Derivatives as Potential DPP IV Inhibitors. The Open Medicinal Chemistry Journal. 2013, 7, 39-48.

 

http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3866624/

 

 

5. Ghassan Shattat, Tariq Al-Qirim, Ghassan Abu Sheikha, Yusuf Al-Hiari, Kamal Sweidan, Rania Al-Qirim, Suhair Hikmat, Lama Hamadneh, Sameer Al-kouz  The Pharmacological Effects of Novel 5-Fluoro-N-(9,10-dihydro-9,10-dioxoanthracen-8-yl)-1H-indole-2-carboxamide Derivatives on Plasma Lipid Profile of Triton-WR-1339-Induced Wistar Rats. Journal of Enzyme Inhibition and Medicinal Chemistry. 2013, 28(4), 863-869.

http://informahealthcare.com/doi/abs/10.3109/14756366.2012.692085

6. Tariq Al-Qirim, Ghassan Shattat, Kamal Sweidan, Waseem El-Huneidi, Ghassan Abu Sheikha, Reema Abu Khalafand Suhair Hikmat. In vivo Antihyperlipidemic Activity of New Series of N- (benzoylphenyl) and N-(acetylphenyl)-1-benzofuran-2- carboxamides in Rats. Archiv der Pharmazie (Weinheim, Germany), 2012, 345(5), 401-406.

 

 

7. Reema Abu Khalaf, Ghassan Abu Sheikha, Ghadeer Albadawi, and Mutasem O. Taha. Design, synthesis and biological evaluation of sulfonic acid ester and benzenesulfonamide derivatives as potential CETP inhibitors. Medicinal Chemistry Research, 2012, 21(11), 3669-3680. http://link.springer.com/article/10.1007%2Fs00044-011-9917-5#page-1

 

 

8. Yusuf Al-Hiari, Ghassan Shattat, Tariq Al-Qirim, Waseem El-Huneidi, Ghassan Abu Sheikha and Suhair Hikmat. Antihyperlipidemic Properties of Novel N-(Benzoylphenyl)-5-substituted-1H-indole-2-carboxamides in     Triton WR-1339-Induced Hyperlipidemic Rats. Molecules 2011, 16(10): 8292-8304.

 

http://www.mdpi.com/1420-3049/16/10/8292

 

 

9. Rana M. OBAIDAT, Ammar BADER , Wafa AL-RAJAB , Ghassan ABU SHEIKHA  , Aiman A. OBAIDAT. Preparation of Mucoadhesive Oral Patches Containing Tetracycline Hydrochloride and Carvacrol for Treatment of Local Mouth Bacterial Infections and Candidiasis. Sci. Pharm. 2011; 79: 197–212.

 

http://www.ncbi.nlm.nih.gov/pubmed/21617783

 

 

10. Ghassan Abu Sheikha, Mahmoud A. Al-Sha’er, Mutasem O. Taha. Some Sulfonamide drugs inhibit ATP-ase activity of heat shock protein 90: investigation by docking   simulation and experimental validation. Journal of Enzyme Inhibition and Medicinal Chemistry, 26, 603-609, 2011.

 

http://informahealthcare.com/doi/abs/10.3109/14756366.2010.541394

 

 

11. Ghassan Abu Sheikha, Buthina Hussin, Yusuf Al-Hiari, Tariq Al-Qirim and Ghassan Shattat. Synthesis of Benzothiophene Carboxamide Derivatives and Their Pharmacological Evaluation as Potent Antihypertriglyceridemic Agents in Rats.  Z. Naturforsch, 66c, 93-103, 2011.

 

http://www.ncbi.nlm.nih.gov/pubmed/21630582

 

 

12. Ghassan Shattat, Rania Al-Qirim, Yusuf Al-Hiari, Ghassan Abu sheikha, Tariq Al-Qirim, Waseem El-Huneidi and Moyad Shahwan. Synthesis and      Anti-Hyperlipidemic Evaluation of N-(Benzoylphenyl)-5-fluoro-1H-indole-2-carboxamide Derivatives in Triton WR-1339-Induced Hyperlipidemic Rats. Molecules 15, 5840-5849, 2010.

 

http://www.mdpi.com/1420-3049/15/9/5840

 

13. Ghassan Abu Sheikha, Reema Abu Khalaf, Areej Melhem and Ghadeer Albadawi. Design, Synthesis, and Biological Evaluation of Benzylamino-Methanone Based Cholestryl Ester Transfer Protein Inhibitors. Molecules 15, 5721-5733, 2010.

 

http://www.mdpi.com/1420-3049/15/8/5721

 For more publications please see C.V

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